Abstract

RISE-IIP: Riociguat for the treatment of pulmonary hypertension associated with idiopathic interstitial pneumonia

Pulmonary hypertension (PH) complicating idiopathic interstitial pneumonias (IIPs) is associated with impaired functional ability and poor outcomes. Whether treating PH in IIP is beneficial remains unknown.

RISE-IIP (NCT02138825) was a randomised, placebo (PBO)-controlled study to evaluate the efficacy and safety of riociguat in patients with IIP, FVC ≥45% predicted and mean pulmonary artery pressure ≥25 mmHg.

Patients were randomised to riociguat up to 2.5 mg tid or PBO for 26 weeks followed by an open-label extension where all patients received riociguat. The primary endpoint was change from baseline to week 26 in 6-minute walk distance (6MWD). Secondary endpoints included clinical worsening (all-cause mortality, hospitalisation due to worsening cardiopulmonary status, 15% decrease in 6MWD or worsening of WHO FC).

Of 147 randomised patients, 73 received riociguat and 74 PBO. The study was stopped early (mean treatment duration 121±66 days) at the recommendation of the Data Monitoring Committee due to increased SAEs (37% riociguat vs 23% PBO in the blinded phase) and increased mortality in riociguat patients. There were 11 deaths in the blinded phase (8 riociguat, 3 PBO), and 9 in the extension (1 former riociguat, 8 former PBO). Riociguat did not improve 6MWD vs PBO at 26 week (least squares mean difference +21 m; 95% CI –9 to +52 m). There was no difference in proportion of subjects with clinical worsening: 47% riociguat vs 49% PBO.

In patients with PH-IIP, riociguat was associated with increased SAEs and mortality, and an unfavourable risk:benefit ratio. The current study did not reveal a potential aetiology for the observed mortality effect.